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Organic Chemistry

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Cheminformatic Analysis of Core-Atom Transformations in Pharmaceutically Relevant Heteroaromatics

G. Logan Bartholomew, Lucas J. Karas, Reilly M. Eason, Charles S. Yeung, Matthew S. Sigman, Richmond Sarpong

Version 1 posted 19 November 2024

981

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Organic Chemistry

Working Paper

Synthesis of Bicyclo[1.1.0]butanes from Iodo-Bicyclo[1.1.1]pentanes

Michael Mandler, James Mignone, Elizabeth Jurica, Maximilian Palkowitz, Darpandeep Aulakh, Anthony Cauley, Christopher Farley, Shasha Zhang, Sarah Traeger, Amy Sarjeant, Anthony Paiva, Heidi Perez, Bruce Ellsworth, Alicia Regueiro-Ren

Version 2 posted 29 May 2023

2,591

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Organic Chemistry

Working Paper

Unified Access to Pyrimidines and Quinazolines Enabled by N-N Cleaving Carbon Atom Insertion

Ethan Hyland, Patrick Kelly, Alexander McKillop, Balu Dherange, Mark Levin

Version 1 posted 09 September 2022

2,144

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Organic Chemistry

Working Paper

Late-stage diversification of indole skeletons through nitrogen atom insertion

Julia C. Reisenbauer, Ori Green, Allegra Franchino, Patrick Finkelstein, Bill Morandi

Version 1 posted 25 May 2022

4,795

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Organic Chemistry

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Carbon-to-nitrogen atom swap enables direct access to benzimidazoles from drug-like indoles

Ann-Sophie Paschke, Yannick Brägger, Bence Botlik, Erich Staudinger, Ori Green, Bill Morandi

Version 1 posted 14 October 2024

3,460

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Inorganic Chemistry

Working Paper

A Synthetic Cycle for Heteroarene Synthesis by Nitride Insertion

Patrick Kelly, Alexander Filatov, Mark Levin

Version 1 posted 07 July 2022

2,508

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Organic Chemistry

Working Paper

Tailoring Unstrained Pyrrolidines via Reductive C–N Bond Cleavage with Lewis Acid and Photoredox Catalysis

Marina Hirao, Kazuhiro Aida, Tsuyoshi Saitoh, Takashi Yamamoto, Yasuaki Einaga, Eisuke Ota, Junichiro Yamaguchi

Version 1 posted 30 July 2024

957

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Organic Chemistry

Working Paper

Electrochemical Single-Carbon Insertion: Unlocking para-Insertion via Distonic Radical Cation Intermediates

Tatsuya Morimoto, Yoshio Nishimoto, Taku Suzuki-Osborne, Su-Gi Chong, Kazuhiro Okamoto, Azusa Kikuchi, Daisuke Yokogawa, Mahito Atobe, Naoki Shida

Version 1 posted 21 October 2024

643

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Organic Chemistry

Working Paper

Accessing Sulfonamides via Formal SO2 Insertion into C–N Bonds

Myojeong Kim, Carys Obertone, Christopher Kelly, Christopher Reiher, Cristina Grosanu, James Robertson, Mark Levin

Version 1 posted 22 August 2024

4,390

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Organic Chemistry

Working Paper

Evidence for Dearomatizing Spirocyclization and Dynamic Effects in the Nitrogen Deletion of Tetrahydroisoquinolines

Jeanne Masson-Makdissi, Remy Lalisse, Mingbin Yuan, Balu Dherange, Osvaldo Gutierrez, Mark Levin

Version 2 posted 20 February 2024

2,571

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20 results in Skeletal editing in Keywords: Skeletal editing

Cheminformatic Analysis of Core-Atom Transformations in Pharmaceutically Relevant Heteroaromatics

Synthesis of Bicyclo[1.1.0]butanes from Iodo-Bicyclo[1.1.1]pentanes

Unified Access to Pyrimidines and Quinazolines Enabled by N-N Cleaving Carbon Atom Insertion

Late-stage diversification of indole skeletons through nitrogen atom insertion

Carbon-to-nitrogen atom swap enables direct access to benzimidazoles from drug-like indoles

A Synthetic Cycle for Heteroarene Synthesis by Nitride Insertion

Tailoring Unstrained Pyrrolidines via Reductive C–N Bond Cleavage with Lewis Acid and Photoredox Catalysis

Electrochemical Single-Carbon Insertion: Unlocking para-Insertion via Distonic Radical Cation Intermediates

Accessing Sulfonamides via Formal SO2 Insertion into C–N Bonds

Evidence for Dearomatizing Spirocyclization and Dynamic Effects in the Nitrogen Deletion of Tetrahydroisoquinolines

20 results in Keywords: Skeletal editing