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Biological and Medicinal Chemistry

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Labeling Preferences of Diazirines with Protein Biomolecules

Alexander West, Giovanni Muncipinto, Hung-Yi Wu, Andrew Huang, Matthew T. Labenski, Christina Woo

Version 1 posted 17 December 2020

1,393

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Biological and Medicinal Chemistry

Working Paper

Discovery of an MLLT1/3 YEATS Domain Chemical Probe

Moses Moustakim, Thomas Christott, Octovia P. Monteiro, James Bennett, Charline Giroud, Jennifer Ward, Catherine Rogers, Paul Smith, Ioanna Panagakou, Laura Diaz Saez, Suet Ling Felce, Vicki Gamble, Carina Gileadi, Nadia Halidi, David Heidenreich, Apirat Chaikuad, Stefan Knapp, Kilian Huber, Gillian Farnie, Jag Heer, Nenad Manevski, Gennady Poda, Rima Al-awar, Darren J. Dixon, Paul E. Brennan, Oleg Fedorov

Version 1 posted 18 September 2018

592

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Biological and Medicinal Chemistry

Working Paper

Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor

Ricardo Serafim, André Santiago, Caio dos Reis, Jessica Takarada, Priscila Mezzomo, Katlin Massirer, Martin P. Schwalm, Mark Kudolo, Stefan Gerstenecker, Apirat Chaikuad, Stefan Knapp, Stefan Laufer, Rafael Counago, Matthias Gehringer

Version 1 posted 20 May 2021

977

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Biological and Medicinal Chemistry

Working Paper

Will the Chemical Probes Please Stand Up?

Ctibor Škuta, Christopher Southan, Petr Bartunek

Version 2 posted 02 July 2021

627

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Biological and Medicinal Chemistry

Working Paper

Probing Cellular Outcomes Using Heterobivalent Constructs

Rohit Bhadoria, Kefeng Ping, Christer Lohk, Ivar Järving, Pavel Starkov

Version 1 posted 22 January 2019

586

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Biological and Medicinal Chemistry

Working Paper

Discovery of a Potent and Highly Isoform-Selective Inhibitor of the Neglected Ribosomal Protein S6 Kinase Beta 2 (S6K2)

Stefan Gerstenecker, Lisa Haarer, Martin Schröder, Mark Kudolo, Martin P. Schwalm, Valentin Wydra, Ricardo Serafim, Apirat Chaikuad, Stefan Knapp, Stefan Laufer, Matthias Gehringer

Version 1 posted 15 July 2021

363

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Biological and Medicinal Chemistry

Working Paper

Microplate-Based Enzymatic Activity Assay Protocol Powered by Activity-Based Probes

Exequiel Porta, Karunakaran Kalesh, Jaime Isern, Patrick Steel

Version 2 posted 16 April 2024

247

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Biological and Medicinal Chemistry

Working Paper

Aza-SAHA Derivatives are Selective Histone Deacetylase 10 Chemical Probes That Inhibit Polyamine Deacetylation and Phenocopy HDAC10 Knockout

Raphael R. Steimbach, Corey J. Herbst-Gervasoni, Severin Lechner, Tracy Murray Stewart, Glynis Klinke, Johannes Ridinger, Magalie Géraldy, Gergely Tihanyi, Jackson R. Foley, Ulrike Uhrig, Bernhard Kuster, Gernot Poschet, Robert A. Casero, Guillaume Médard, Ina Oehme, David W. Christianson, Nikolas Gunkel, Aubry K. Miller

Version 2 posted 12 May 2022

892

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Biological and Medicinal Chemistry

Working Paper

Piperazine-fused cyclic disulfides: high-performance bioreduction-activated cores for bifunctional probes and reagents

Lukas Zeisel, Jan G. Felber, Karoline C. Scholzen, Carina Schmitt, Alexander J. Wiegand, Leonid Komissarov, Elias S. J. Arnér, Oliver Thorn-Seshold

Version 2 posted 10 October 2023

1,110

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Organic Chemistry

Working Paper

Stereoselective Synthesis of Allele-Specific BET Inhibitors

Adam Bond, Andrea Testa, Alessio Ciulli

Version 1 posted 18 May 2020

598

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11 results in chemical probes in Keywords: chemical probes

Labeling Preferences of Diazirines with Protein Biomolecules

Discovery of an MLLT1/3 YEATS Domain Chemical Probe

Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor

Will the Chemical Probes Please Stand Up?

Probing Cellular Outcomes Using Heterobivalent Constructs

Discovery of a Potent and Highly Isoform-Selective Inhibitor of the Neglected Ribosomal Protein S6 Kinase Beta 2 (S6K2)

Microplate-Based Enzymatic Activity Assay Protocol Powered by Activity-Based Probes

Aza-SAHA Derivatives are Selective Histone Deacetylase 10 Chemical Probes That Inhibit Polyamine Deacetylation and Phenocopy HDAC10 Knockout

Piperazine-fused cyclic disulfides: high-performance bioreduction-activated cores for bifunctional probes and reagents

Stereoselective Synthesis of Allele-Specific BET Inhibitors

11 results in Keywords: chemical probes