Search

Organic Chemistry

Working Paper

Reductive Cleavage of Secondary Sulfonamides: Converting Terminal Functional Groups into Versatile Synthetic Handles

Patrick Fier, Suhong Kim, Kevin M. Maloney

Version 1 posted 03 October 2019

925

Downloads

Organic Chemistry

Working Paper

Remote Formation of Arynes via Formal Dehydrogenation of Arenes

Riley Roberts, Bryan Metze, Aleksandra Nilova, David Stuart

Version 1 posted 25 August 2022

822

Downloads

Organic Chemistry

Working Paper

3-Selective Halogenation of Pyridines via Zincke Imine Intermediates

Benjamin T. Boyle, Jeffrey N. Levy, Louis de Lescure, Robert S. Paton, Andrew McNally

Version 3 posted 12 July 2022

3,631

Downloads

1

Citations

Theoretical and Computational Chemistry

Working Paper

Enabling late-stage drug diversification by high-throughput experimentation with geometric deep learning

David F. Nippa, Kenneth Atz, Remo Hohler, Alex T. Müller, Andreas Marx, Christian Bartelmus, Georg Wuitschik, Irene Marzuoli, Vera Jost, Jens Wolfard, Martin Binder, Antonia F. Stepan, David B. Konrad, Uwe Grether, Rainer E. Martin, Gisbert Schneider

Version 2 posted 15 November 2022

2,661

Downloads

3

Citations

Theoretical and Computational Chemistry

Working Paper

Graph transformer neural network for chemical reactivity prediction

David F. Nippa, Kenneth Atz, Alex T. Müller, Jens Wolfard, Clemens Isert, Martin Binder, Oliver Scheidegger, David B. Konrad, Uwe Grether, Rainer E. Martin, Gisbert Schneider

Version 1 posted 16 May 2023

1,287

Downloads

Organic Chemistry

Working Paper

Engineering Central Substitutions in Heptamethine Dyes via Aryl-lithium Addition for Improved Fluorophore Performance

Lei Guo, Meek Yang, Bin Dong, Seth Lewman, Alex Van Horn, Shang Jia

Version 1 posted 27 March 2024

457

Downloads

Catalysis

Working Paper

Ruthenium-catalysed C‒H amidation for the late-stage synthesis of PROTACs

Daniele Antermite, Stig D. Friis, Johan R. Johansson, Okky D. Putra, Lutz Ackermann, Magnus J. Johansson

Version 1 posted 27 March 2023

1,087

Downloads

Organic Chemistry

Working Paper

Direct C3-functionalization of indoles with alpha-heteroaryl-substituted methyl alcohols via a metal-free hydrogen autotransfer-type reaction

Ethan Pazur, Nikhil Tasker, Peter Wipf

Version 2 posted 18 October 2023

889

Downloads

Organic Chemistry

Working Paper

A Broadly Applicable Strategy to Aminate Azines Enabled by Electronically Tuned Phosphine Reagents.

Ren-Rong Liu, Jeffrey N. Levy, Andrew McNally

Version 1 posted 08 August 2024

369

Downloads

Organic Chemistry

Working Paper

Late-Stage C(sp2)–C(sp3) Diversification via Nickel Oxidative Addition Complexes

Ruben Martin, Carlota Odena, Maria Lourdes Linares, Nahury Castellanos-Blanco, Ryan McGuire, Jose Manuel Alonso, Alejandro Dieguez, Eric Tan, Jesus Alcazar, Peter Buijnsters, Santiago Cañellas

Version 1 posted 08 August 2023

1,696

Downloads

1

Citations

Refine Search

35 results in Late-Stage Functionalization in Keywords: Late-Stage Functionalization

Reductive Cleavage of Secondary Sulfonamides: Converting Terminal Functional Groups into Versatile Synthetic Handles

Remote Formation of Arynes via Formal Dehydrogenation of Arenes

3-Selective Halogenation of Pyridines via Zincke Imine Intermediates

Enabling late-stage drug diversification by high-throughput experimentation with geometric deep learning

Graph transformer neural network for chemical reactivity prediction

Engineering Central Substitutions in Heptamethine Dyes via Aryl-lithium Addition for Improved Fluorophore Performance

Ruthenium-catalysed C‒H amidation for the late-stage synthesis of PROTACs

Direct C3-functionalization of indoles with alpha-heteroaryl-substituted methyl alcohols via a metal-free hydrogen autotransfer-type reaction

A Broadly Applicable Strategy to Aminate Azines Enabled by Electronically Tuned Phosphine Reagents.

Late-Stage C(sp2)–C(sp3) Diversification via Nickel Oxidative Addition Complexes

35 results in Keywords: Late-Stage Functionalization