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Abstract
The regiospecific ring expansion of 2H-azetines into halogenated pyrroles is disclosed. Simple reaction sequences have been developed to conceptualize this 4-to-5 skeletal editing strategy, taking advantage of the inherent reactivity of double bonds present in the initial four-membered ring systems. Such reaction design allows for the preparation of highly substi-tuted halogenated pyrrole derivatives.
Supplementary materials
Title
Supporting information for "Regiospecific Skeletal Editing of Azetines towards Halogenated Pyrroles"
Description
Contains all methods, compound description, 1H- 13C- and 19F-NMR spectra, MS and HRMS data
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